US3314852A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Method of producing ataraxic, anticonvulsant activity and skeletal muscle relaxation
Assignee: Bristol Myers Co
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Filing: 1963-10-04
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Granted: 1967-04-18
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Expires: 1983-10-04
Abstract
No abstract record available.
Inventors
- 👤 Daniel M Green
- 👤 Russell F Krueger
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-01 12:55
CPC Classifications
A; A61; A61K; A61K31/00; A61K31/33; A61K31/395; A61K31/435; A61K31/44; A61K31/21; A61K31/27; A61K31/38; A61K31/41; A61K31/42; A61K31/495; A61K31/505
Claims Analysis
Total Claims: 2
Claim 1
Independent Claim
179 words
A METHOD OF (A) INDUCING RELAXATION OF AT LEAST ONE OF SKELETAL MUSCLE IN ANIMALS SUFFERING FROM INVOLUNTARY CONTRACTIONS OF SKELETAL MUSCLE; AND (B) RELIEVING CONVULSIONS IN AN ANIMAL SUFFERING FROM THE SAME; AND (C) INDUCING ATARAXIA IN AN ANIMAL SUFFERING FROM NERVOUS TENSION; WHICH COMPRISES ORALLY ADMINISTERING TO SAID ANIMAL A THERAPEUTICALLY EFFECTIVE QUANTITY OF THE COMBINATION OF A SKELETAL MUSCLE RELAXANT AND AN ANTIHISTAMINE OR A PAHARMACEUTICALLY ACCEPTABLE NON-TOXIC ACID ADDITION SALT THEREOF IN THE RATIO OF 4 TO 32 PARTS OF SKELETAL MUSCLE RELAXANT PER PART OF ANTIHISTAMINE; SAID MUSCLE RELAXANT BEING SELECTED FROM THE GROUP CONSISTING OF GLYCERYL GUAIACOLATE, METHOCARBAMOYL, MEPHENESIN, MEPHENESIN CARBAMATE, CARIOPRODOL, EMYLCAMATE, MEPROBAMATE, HYDROXYPHENAMATE, STYRAMATE, CHLORZOXAZONE, ZOXAZOLAMINE, HYDROXYZINE AND PHENAGLYCODOL;L AND SAID ANTIHISTAMINE BEING SELECTED FROM THE GROUP CONSISTING OF TRIPELENNAMINE HCL, PYRILAMINE MALEATE, THONZYLAMINE HCL, METAPHENILENE HCL, METHJAPYRILENE HCL, CHLOROTHEN CITRATE, THENYLDIAMINE HCL, MECLIZINE HYDROCHLORIDE, CYCLIZINE HYDROCHLORIDE, CLORCYCLIZINE, PROMETHAZINE HYDROCHLORIDE, PYRATHIAZINE HYDROCHLORIDE, PHENIRAMINE MALEATE, CHLORPHENIRAMINE MALEATE, BROMMPHENIRAMINE MALEATE (D-ISOMER), TRIPROLIDONE HYDROCHLORIDE, PYRROBUTAMINE PHOSPHATE, DIPHENYLPYRALINE HYDROCHLORIDE, PHENINDAMINE TARTRATE, DIPHENHYDRAMINE, DIMENHYDRINATE, BROMODIPHENHYDRAMINE, DOXYLAMINE SUCCINATE, CARBINOXAMINE MALEATE, PHENYLLTOLOXAMINE DIHYDROGEN CITRATE AND PHENYLTOLOXAMINE DIHYDROGEN HYDROCHLORIDE.
Claim 2
Independent Claim
179 words
A METHOD OF (A) INDUCING RELAXATION OF AT LEAST ONE OF SKELETAL MUSCLE IN ANIMALS SUFFERING FROM INVOLUNTARY CONTRACTIONS OF SKELETAL MUSCLE; AND (B) RELIEVING CONVULSIONS IN AN ANIMAL SUFFERING FROM THE SAME; AND (C) INDUCING ATARAXIA IN AN ANIMAL SUFFERING FROM NERVOUS TENSION; WHICH COMPRISES ORALLY ADMINISTERING TO SAID ANIMAL A THERAPEUTICALLY EFFECTIVE QUANTITY OF THE COMBINATION OF A SKELETAL MUSCLE RELAXANT AND AN ANTIHISTAMINE OR A PAHARMACEUTICALLY ACCEPTABLE NON-TOXIC ACID ADDITION SALT THEREOF IN THE RATIO OF 4 TO 32 PARTS OF SKELETAL MUSCLE RELAXANT PER PART OF ANTIHISTAMINE; SAID MUSCLE RELAXANT BEING SELECTED FROM THE GROUP CONSISTING OF GLYCERYL GUAIACOLATE, METHOCARBAMOYL, MEPHENESIN, MEPHENESIN CARBAMATE, CARIOPRODOL, EMYLCAMATE, MEPROBAMATE, HYDROXYPHENAMATE, STYRAMATE, CHLORZOXAZONE, ZOXAZOLAMINE, HYDROXYZINE AND PHENAGLYCODOL;L AND SAID ANTIHISTAMINE BEING SELECTED FROM THE GROUP CONSISTING OF TRIPELENNAMINE HCL, PYRILAMINE MALEATE, THONZYLAMINE HCL, METAPHENILENE HCL, METHJAPYRILENE HCL, CHLOROTHEN CITRATE, THENYLDIAMINE HCL, MECLIZINE HYDROCHLORIDE, CYCLIZINE HYDROCHLORIDE, CLORCYCLIZINE, PROMETHAZINE HYDROCHLORIDE, PYRATHIAZINE HYDROCHLORIDE, PHENIRAMINE MALEATE, CHLORPHENIRAMINE MALEATE, BROMMPHENIRAMINE MALEATE (D-ISOMER), TRIPROLIDONE HYDROCHLORIDE, PYRROBUTAMINE PHOSPHATE, DIPHENYLPYRALINE HYDROCHLORIDE, PHENINDAMINE TARTRATE, DIPHENHYDRAMINE, DIMENHYDRINATE, BROMODIPHENHYDRAMINE, DOXYLAMINE SUCCINATE, CARBINOXAMINE MALEATE, PHENYLLTOLOXAMINE DIHYDROGEN CITRATE AND PHENYLTOLOXAMINE DIHYDROGEN HYDROCHLORIDE.
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USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1970-04-17 | 1970-10-17 | 1971-04-18 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1974-04-17 | 1974-10-17 | 1975-04-18 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1978-04-17 | 1978-10-17 | 1979-04-18 | $7700.00 | Window Closed / Lapsed |