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US3681340A Expired / Lapsed US ⏱️ 0.0 years remaining

1,3-benzodiazepines

Assignee: Individual
•
Filing: 1968-02-12
•
Granted: 1972-08-01
•
Expires: 1988-02-12
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Abstract

Abstract 4,5-Dihydro-3H-1,3-benzodiazepines, e.g., those of the formula N-oxides, quaternaries and salts thereof exhibit central nervous system depressing and coronary dilatating effects.

Inventors

  • 👤 Herman Robert Rodriguez
  • 👤 George De Stevens

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-01 22:12
CPC Classifications
C; C07; C07D; C07D333/00; C07D333/02; C07D333/04; C07D333/26; C07D333/38

Claims Analysis

Total Claims: 3
Claim 1
Independent Claim 59 words
A compound as claimed in claim 1, and having the formula in which R10 is amino, methyl, chloromethyl, methoxymethyl, dimethylaminomethyl, piperidinomethyL, 4-phenyl-piperazinomethyl, benzyl, mono- or dimethoxy-benzyl, 2-imidazolylmethyl, phenyl, mono- or dimethyl-phenyl, i-propyl-phenyl, hydroxy-phenyl, mono-, di or trimethoxy-phenyl, ethoxy-phenyl, fluoro-phenyl, chloro-phenyl, trifluoromethyl-phenyl, nitro-phenyl, carboxy-phenyl, carbethoxy-phenyl or dimethylsulfamoyl-phenyl, R11 is hydrogen or methyl, or a therapeutically acceptable acid addition salt thereof.
Claim 2
Dependent Claim 35 words
A compound as claimed in claim 2, in which formula R10 is methyl, piperidinomethyl, benzyl, 4-methoxy-benzyl, phenyl, 4-methoxy-phenyl, 3- or 4-nitro-phenyl or 3-carboxy-phenyl and R11 is hydrogen, or a therapeutically acceptable acid addition salt thereof.
Claim 3
Dependent Claim 19 words
A compound as claimed in claim 1 and being the 2-(3-nitro-phenyl)-7,8-dimethoxy-4,5-dihydro-3H-1,3-benzodiazepine or a therapeutically acceptable acid addition salt thereof.

References Cited (Backward Citations)

US3474090A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1975-08-01 1976-01-31 1976-08-01 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1979-08-01 1980-01-31 1980-08-01 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1983-08-01 1984-01-31 1984-08-01 $7700.00 Window Closed / Lapsed

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