US4100270A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Antibacterial oral composition
Assignee: Colgate Palmolive Co
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Filing: 1977-04-25
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Granted: 1978-07-11
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Expires: 1997-04-25
Abstract
Abstract An antibacterial oral composition effective to promote oral hygiene containing an antibacterial antiplaque agent and an additive which reduces staining of dental surfaces without substantially diminishing the antibacterial and antiplaque activity of the agent. Bis-biguanido hexanes, such as chlorhexidine and alexidine, and quaternary ammonium salts, such as benzethonium chloride and cetyl pyridinium chloride, are typical examples of antibacterial agents. The antistain additive is a polymeric polyphosphonic compound, such as polyallyl bis-(phosphonomethylene) amine acid and salts thereof.
Inventors
- 👤 Abdul Gaffar
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-02 04:00
CPC Classifications
A; A61; A61Q; A61Q11/00; A61K; A61K8/00; A61K8/18; A61K8/30; A61K8/40; A61K8/41; A61K8/416; A61K8/43; A61K8/55; A61K8/72; A61K8/81; A61K8/817; A61K2800/00; A61K2800/40; A61K2800/52
Claims Analysis
Total Claims: 13
Claim 1
Independent Claim
107 words
An oral composition comprising an oral vehicle, a nitrogen containing antibacterial antiplaque agent tending to stain dental surfaces selected from the group consisting of cationic antibacterial antiplaque agent and long chain amine antibacterial antiplaque agent containing a fatty alkyl group of 12 to 18 carbon atoms and a water soluble polymeric polyphosphonic compound antistain additive having the recurring group: ##STR15## wherein X is selected from the group consisting of hydrogen and an orally acceptably action and Y is selected from the group consisting of hydrogen and CH 3 , and the unphosphonated recurring groups of said compound have a total molecular weight of at least about 3,500.
Claim 2
Dependent Claim
107 words
An oral composition comprising an oral vehicle, a nitrogen containing antibacterial antiplaque agent tending to stain dental surfaces selected from the group consisting of cationic antibacterial antiplaque agent and long chain amine antibacterial antiplaque agent containing a fatty alkyl group of 12 to 18 carbon atoms and a water soluble polymeric polyphosphonic compound antistain additive having the recurring group: ##STR15## wherein X is selected from the group consisting of hydrogen and an orally acceptably action and Y is selected from the group consisting of hydrogen and CH 3 , and the unphosphonated recurring groups of said compound have a total molecular weight of at least about 3,500.
Claim 3
Dependent Claim
31 words
The oral composition of claim 1 wherein Y is CH 3 , the molecular weight of the unphosphonated polymer is about 50,000 and the degree of phosphonation is about 15 16%.
Claim 4
Dependent Claim
50 words
The oral composition of claim 1 wherein said anti-bacterial antiplaque agent is present in amount to provide about 0.001% to about 15% by weight based on the free base form of said agent and said polymeric polyphosphonic compound is present in amount of about 0.01% to about 10% by weight.
Claim 5
Dependent Claim
46 words
The oral composition of claim 3 wherein said anti-bacterial antiplaque agent is present in amount of about 0.01% to about 5% by weight based on the free base form of said agent and said polymeric polyphosphonic compound is present in a molar excess to said agent.
Claim 6
Dependent Claim
15 words
The oral composition of claim 3 wherein said anti-bacterial antiplaque agent is a substituted guanidine.
Claim 7
Dependent Claim
30 words
The oral composition of claim 5 wherein said antibacterial antiplaque agent is a pharamaceutically acceptable water soluble salt of an agent selected from the group consisting of chlorhexidine and alexidine.
Claim 8
Dependent Claim
20 words
The oral composition of claim 6 wherein said antibacterial antiplaque agent is a pharmaceutically acceptable water soluble salt of chlorhexidine.
Claim 9
Dependent Claim
14 words
The oral composition of claim 3 wherein said antibacterial antiplaque agent is benzethonium chloride.
Claim 10
Dependent Claim
28 words
The oral composition of claim 3 wherein said antibacterial antiplaque agent is a quaternary ammonium compound containing 1 to 2 alkyl groups of 8 to 20 carbon atoms.
Claim 11
Dependent Claim
15 words
The oral composition of claim 9 wherein said antibacterial antiplaque agent is cetyl pyridinium chloride.
Claim 12
Dependent Claim
26 words
The oral composition of claim 1 wherein said vehicle is an aqueous-alcohol and said composition is a mouthwash of pH of about 4.5 to about 10.
Claim 13
Dependent Claim
39 words
The oral composition of claim 1 wherein said vehicle comprises a liquid vehicle and a gelling agent and a dentally acceptable polishing material is present and said composition is a toothpaste of pH of about 4.5 to about 10.
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USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1981-07-10 | 1982-01-09 | 1982-07-11 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1985-07-10 | 1986-01-09 | 1986-07-11 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1989-07-10 | 1990-01-09 | 1990-07-11 | $7700.00 | Window Closed / Lapsed |