US4153707A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Fungicidal isoxazolyl phenols and method of use
Assignee: Pharmacia and Upjohn Co
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Filing: 1977-11-10
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Granted: 1979-05-08
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Expires: 1997-11-10
Abstract
Abstract A compound of the formula: ##STR1## wherein X is a member selected from the group consisting of hydrogen, alkyl of from 1 to 3 carbon atoms, inclusive, chlorine or bromine; Y is a member selected from the group consisting of hydrogen, chlorine or bromine and R is a member selected from the group consisting of hydrogen or lower alkyl of from 1 to 3 carbon atoms. The compounds can be applied to seeds, plants, animals, objects, or places for preventing damage due to fungi. General methods for preparing the active compounds, compositions and methods of use are shown.
Inventors
- 👤 Malcolm W. Moon
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-10-30 11:48
CPC Classifications
C; C07; C07D; C07D311/00; C07D311/02; C07D311/04; C07D311/22; A; A01; A01N; A01N43/00; A01N43/72; A01N43/80; C07C; C07C45/00; C07C45/45; C07C45/46; C07C45/51; C07C45/54; C07C49/00; C07C49/76; C07C49/82; C07C49/825; C07D261/00; C07D261/02; C07D261/06; C07D261/08
Claims Analysis
Total Claims: 33
Claim 1
Independent Claim
67 words
A compound of the formula: ##STR4## wherein X is a member selected from the group consisting of hydrogen, alkyl of from 1 to 3 carbon atoms, inclusive, chlorine or bromine; Y is a member selected from the group consisting of hydrogen, chlorine or bromine and R is a member selected from the group consisting of hydrogen or lower alkyl of from 1 to 3 carbon atoms, inclusive.
Claim 2
Dependent Claim
67 words
A compound of the formula: ##STR4## wherein X is a member selected from the group consisting of hydrogen, alkyl of from 1 to 3 carbon atoms, inclusive, chlorine or bromine; Y is a member selected from the group consisting of hydrogen, chlorine or bromine and R is a member selected from the group consisting of hydrogen or lower alkyl of from 1 to 3 carbon atoms, inclusive.
Claim 3
Dependent Claim
9 words
A compound according to claim 1 which is 2,4-dichloro-6-(4-methyl-5-isoxazolyl)phenol.
Claim 4
Dependent Claim
9 words
A compound according to claim 1 which is 2,4-dichloro-6-(4-ethyl-5-isoxazolyl)phenol.
Claim 5
Dependent Claim
9 words
A compound according to claim 1 which is 2,4-dibromo-6-(4-methyl-5-isoxazolyl)phenol.
Claim 6
Dependent Claim
9 words
A compound according to claim 1 which is 2-chloro-6-(4-methyl-5-isoxazolyl)phenol.
Claim 7
Dependent Claim
9 words
A compound according to claim 1 which is 2-(4-methyl-5-isoxazolyl)phenol.
Claim 8
Dependent Claim
9 words
A compound according to claim 1 which is 4-methyl-2-(4-methyl-5-isoxazolyl)phenol.
Claim 9
Dependent Claim
9 words
A compound according to claim 1 which is 4-chloro-2-(4-methyl-5-isoxazolyl)phenol.
Claim 10
Dependent Claim
9 words
A compound according to claim 1 which is 2,4-dichloro-6-(5-isoxazolyl)phenol.
Claim 11
Dependent Claim
9 words
A compound according to claim 1 which is 4-chloro-2-(5-isoxazolyl)phenol.
Claim 12
Independent Claim
87 words
A method for controlling fungi comprising the application of an effective antifungal amount of a compound of the formula: ##STR5## wherein X is a member selected from the group consisting of hydrogen, alkyl of from 1 to 3 carbon atoms, inclusive, chlorine or bromine; Y is a member selected from the group consisting of hydrogen, chlorine or bromine and R is a member selected from the group consisting of hydrogen or lower alkyl of from 1 to 3 carbon atoms, inclusive, to fungi, objects or a situs.
Claim 13
Independent Claim
87 words
A method for controlling fungi comprising the application of an effective antifungal amount of a compound of the formula: ##STR5## wherein X is a member selected from the group consisting of hydrogen, alkyl of from 1 to 3 carbon atoms, inclusive, chlorine or bromine; Y is a member selected from the group consisting of hydrogen, chlorine or bromine and R is a member selected from the group consisting of hydrogen or lower alkyl of from 1 to 3 carbon atoms, inclusive, to fungi, objects or a situs.
Claim 14
Dependent Claim
9 words
A method according to claim 11 which is 2,4-dichloro-6-(4-methyl-5-isoxazolyl)phenol.
Claim 15
Dependent Claim
9 words
A method according to claim 11 which is 2,4-dichloro-6-(4-ethyl-5-isoxazolyl)phenol.
Claim 16
Dependent Claim
9 words
A method according to claim 11 which is 2,4-dibromo-6-(4-methyl-5-isoxazolyl)phenol.
Claim 17
Dependent Claim
9 words
A method according to claim 11 which is 2-chloro-6-(4-methyl-5-isoxazolyl)phenol.
Claim 18
Dependent Claim
9 words
A method according to claim 11 which is 2-(4-methyl-5-isoxazolyl)phenol.
Claim 19
Dependent Claim
9 words
A method according to claim 11 which is 4-methyl-2-(4-methyl-6-isoxazolyl)phenol.
Claim 20
Dependent Claim
9 words
A method according to claim 11 which is 4-chloro-2-(4-methyl-5-isoxazolyl)phenol.
Claim 21
Dependent Claim
9 words
A method according to claim 11 which is 2,4-dichloro-6-(5-isoxazolyl)phenol.
Claim 22
Dependent Claim
9 words
A method according to claim 11 which is 4-chloro-2-(5-isoxazolyl)phenol.
Claim 23
Dependent Claim
81 words
A composition comprising a fungicidal amount of a pg,27 compound of the formula: ##STR6## wherein X is a member selected from the group consisting of hydrogen, alkyl of from 1 to 3 carbon atoms, inclusive, chlorine or bromine; Y is a member selected from the group consisting of hydrogen, chlorine or bromine and R is a member selected from the group consisting of hydrogen or lower alkyl of from 1 to 3 carbon atoms, inclusive, in association with an inert carrier.
Claim 24
Dependent Claim
81 words
A composition comprising a fungicidal amount of a pg,27 compound of the formula: ##STR6## wherein X is a member selected from the group consisting of hydrogen, alkyl of from 1 to 3 carbon atoms, inclusive, chlorine or bromine; Y is a member selected from the group consisting of hydrogen, chlorine or bromine and R is a member selected from the group consisting of hydrogen or lower alkyl of from 1 to 3 carbon atoms, inclusive, in association with an inert carrier.
Claim 25
Dependent Claim
9 words
A composition according to claim 21 which is 2,4-dichloro-6-(4-methyl-5-isoxazolyl)phenol.
Claim 26
Dependent Claim
9 words
A composition according to claim 21 which is 2,4-dichloro-6-(4-ethyl-5-isoxazolyl)phenol.
Claim 27
Dependent Claim
9 words
A composition according to claim 21 which is 2,4-dibromo-6-(4-methyl-5-isoxazolyl)phenol.
Claim 28
Dependent Claim
9 words
A composition according to claim 21 which is 2-chloro-6-(4-methyl-5-isoxazolyl)phenol.
Claim 29
Dependent Claim
9 words
A composition according to claim 21 which is 2-(4-methyl-5-isoxazolyl)phenol.
Claim 30
Dependent Claim
9 words
A composition according to claim 21 which is 4-methyl-2-(4-methyl-5-isoxazolyl)phenol.
Claim 31
Dependent Claim
9 words
A composition according to claim 21 which is 4-chloro-2-(4-methyl-5-isoxazolyl)phenol.
Claim 32
Dependent Claim
9 words
A composition according to claim 21 which is 2,4-dichloro-6-(5-isoxazolyl)phenol.
Claim 33
Dependent Claim
9 words
A composition according to claim 21 which is 4-chloro-2-(5-isoxazolyl)phenol.
References Cited (Backward Citations)
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1982-05-07 | 1982-11-06 | 1983-05-08 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1986-05-07 | 1986-11-06 | 1987-05-08 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1990-05-07 | 1990-11-06 | 1991-05-08 | $7700.00 | Window Closed / Lapsed |