US4160838A
Expired / Lapsed
US
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Antimicrobial and plant-growth-regulating triazole derivatives
Assignee: Janssen Pharmaceutica NV
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Filing: 1978-01-03
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Granted: 1979-07-10
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Expires: 1998-01-03
Abstract
Abstract Novel 1-(β-aryl)ethyl-1H-1,2,4-triazole ketals useful for their antimicrobial and plant-growth regulating activities.
Inventors
- 👤 Gustaaf Van Reet
- 👤 Jan Heeres
- 👤 Lourens Wals
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-06 08:44
CPC Classifications
C; C07; C07D; C07D231/00; C07D231/02; C07D231/10; C07D231/12; A; A01; A01N; A01N43/00; A01N43/64; A01N43/647; A01N43/653; C07D233/00; C07D233/54; C07D233/56; C07D249/00; C07D249/02; C07D249/08; C07D317/00; C07D317/08; C07D317/10; C07D317/14; C07D317/16; C07D317/18; C07D317/22; C07D317/30
Claims Analysis
Total Claims: 14
Claim 1
Independent Claim
145 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of a 1-(β-aryl)ethyl-1H-1,2,4-triazole ketal of the formula: ##STR9## and the therapeutically active acid addition salts thereof, wherein: Z is an alkylene selected from the group consisting of --CH 2 --CH 2 --, --CH 2 --CH 2 --CH 2-- , --CH(CH 3 )--CH(CH 3 )--and --CH 2 --CH(alkyl)--, wherein said alkyl has from 1 to 10 carbon atoms; and Ar is a member selected from the group consisting of phenyl, substituted phenyl, thienyl, 5-chloro-2-thienyl, naphthyl, fluorenyl, and wherein "substituted phenyl" has the meaning of a phenyl radical having thereon from 1 to 3 substituents selected independently from the group consisting of halo, lower alkyl, lower alkyloxy, cyano and nitro.
Claim 2
Dependent Claim
145 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of a 1-(β-aryl)ethyl-1H-1,2,4-triazole ketal of the formula: ##STR9## and the therapeutically active acid addition salts thereof, wherein: Z is an alkylene selected from the group consisting of --CH 2 --CH 2 --, --CH 2 --CH 2 --CH 2-- , --CH(CH 3 )--CH(CH 3 )--and --CH 2 --CH(alkyl)--, wherein said alkyl has from 1 to 10 carbon atoms; and Ar is a member selected from the group consisting of phenyl, substituted phenyl, thienyl, 5-chloro-2-thienyl, naphthyl, fluorenyl, and wherein "substituted phenyl" has the meaning of a phenyl radical having thereon from 1 to 3 substituents selected independently from the group consisting of halo, lower alkyl, lower alkyloxy, cyano and nitro.
Claim 3
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 4
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 5
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4-methyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 6
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4-methyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 7
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4-ethyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 8
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4-ethyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 9
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4-propyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 10
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4-propyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 11
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4-pentyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 12
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4-pentyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 13
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4,5-dimethyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
Claim 14
Dependent Claim
47 words
A composition for combatting a microorganism selected from the group consisting of fungus and bacterium comprising an inert carrier material and as an active ingredient an effective amount of a chemical compound selected from the group consisting of 1-[2-(2,4-dichlorophenyl)-4,5-dimethyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole and the therapeutically active acid addition salts thereof.
References Cited (Backward Citations)
DE2551560A1
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1982-07-09 | 1983-01-08 | 1983-07-10 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1986-07-09 | 1987-01-08 | 1987-07-10 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1990-07-09 | 1991-01-08 | 1991-07-10 | $7700.00 | Window Closed / Lapsed |