US4340539A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Derivatives of 6-bromo penicillanic acid
Assignee: Bristol Myers Co
•
Filing: 1980-12-11
•
Granted: 1982-07-20
•
Expires: 2000-12-11
Abstract
Abstract 2β-Chloromethyl-2α-methylpenam-3α-carboxylic acid sulfone and salts and esters thereof were synthesized and found to be potent inhibitors of β-lactamases.
Inventors
- 👤 William J. Gottstein
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-10-24 22:22
CPC Classifications
C; C07; C07D; C07D499/00
Claims Analysis
Total Claims: 9
Claim 1
Independent Claim
12 words
An ester having the formula ##STR59## wherein R is benzyl or p-nitrobenzyl.
Claim 2
Dependent Claim
12 words
An ester having the formula ##STR59## wherein R is benzyl or p-nitrobenzyl.
Claim 3
Dependent Claim
9 words
The ester of claim 1 wherein R is p-nitrobenzyl.
Claim 4
Dependent Claim
13 words
An ester having the formula ##STR60## wherein R is benzyl, p-nitrobenzyl or β,β,β-trichloroethyl.
Claim 5
Dependent Claim
13 words
An ester having the formula ##STR60## wherein R is benzyl, p-nitrobenzyl or β,β,β-trichloroethyl.
Claim 6
Dependent Claim
9 words
The ester of claim 3 wherein R is p-nitrobenzyl.
Claim 7
Dependent Claim
9 words
The ester of claim 3 wherein R is β,β,β-trichloroethyl.
Claim 8
Dependent Claim
6 words
The ester having the formula ##STR61##
Claim 9
Dependent Claim
6 words
The ester having the formula ##STR61##
References Cited (Backward Citations)
US3197466A
Cited
GB1072108A
Cited
US3544581A
Cited
US3867538A
Cited
US3536698A
Cited
US3697507A
Cited
US3954735A
Cited
US3873521A
Cited
US3869449A
Cited
US3951954A
Cited
US3963704A
Cited
US3860579A
Cited
US4036829A
Cited
US3939180A
Cited
US4036847A
Cited
US3993646A
Cited
US4009159A
Cited
US3928595A
Cited
US3941774A
Cited
US3989685A
Cited
US3954732A
Cited
US3996236A
Cited
US3931150A
Cited
US4046759A
Cited
US4058521A
Cited
US4181659A
Cited
US4081546A
Cited
US4155912A
Cited
US4180506A
Cited
US4203993A
Cited
US4203992A
Cited
US4217274A
Cited
GB2044255A
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1985-07-19 | 1986-01-18 | 1986-07-20 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1989-07-19 | 1990-01-18 | 1990-07-20 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1993-07-19 | 1994-01-18 | 1994-07-20 | $7700.00 | Window Closed / Lapsed |