Claims Analysis
Total Claims: 12
Claim 1
Independent Claim
363 words
A compound of the formulae I or II ##STR32## in which A is a radical of the formulae III, IV or V ##STR33## R 1 and R 4 are --H or --Cl, R 2 and R 5 are --H, halogen, --NO 2 , --CN, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, --CF 3 or phenyloxy which is unsubstituted or substituted by one or two chlorine atoms, one or two methyl or methoxy groups, or by one or two chlorine atoms and one or two methyl or methoxy groups and R 3 is alkyl having at least 10 C atoms, X is a radical of the formulae --NH--, --O--, ##STR34## n is the number 1 or 2, Y is the radical of the formulae --COO--, --OOC--, --CONH-- or --NHCO-- or a radical of the formulae ##STR35## in which R 1 and R 2 are as defined above, D is a 5-benzimidazolonyl, 5- or 6-benzoxazolonyl, 6-(2,4-dihydroxy)-quinazolinyl, 6- or 7-(4-methyl)quinolone-2-yl, 6- or 7-phenmorpholone-3-yl or 6-quinazolone-4-yl radical, Z is --H, --Br, --OCH 3 , --CN or --NO 2 and X 1 , and X 2 , independently of one another, are --H, halogen, --CH 3 , --OCH 3 --OC 2 H 5 or --NO 2 and X 3 is --H, --NHCO--C 1 -C 4 -alkyl, benzoylamino or phenylcarboxamido which are each unsubstituted or substituted on the phenyl ring by one or two chlorine atoms, one or two methyl or methoxy groups, one or two chlorine atoms and one or two methyl or methoxy groups, or an --NHCO--C 1 -C 4 alkyl group, or X 2 and X 3 together with the carbon atom to which they are bound are an aromatic carboxylic 6-membered ring or an aromatic heterocyclic 5- or 6-membered ring selected from the group consisting of 5-amino-benzimidazolone, 7-chloro-5-amino-benzimidazolone, 7-bromo-5-amino-benzimidazolone, 6-chloro-5-amino-benzimidazolone, 6-bromo-5-amino-benzimidazolone, 6-methoxy-5-amino-benzimidazolone, 7-methoxy-5-amino-benzimidazolone, 6-ethoxy-5-amino-benzimidazolone, 7-chloro-4-methyl-5-amino-benzimidazolone, 6-methyl-5-amino-benzimidazolone, 4,7-dimethyl-5-amino-benzimidazolone, 4-methyl-6-chloro-5-amino-benzimidazolone, 5-amino-1-methyl-benzimidazolone, 6-amino-2,4-dihydroxyquinazoline, 6-amino-1,4-dihydroxyquinazoline, 6-amino-4-methyl-2-quinolone, 7-amino-4-methyl-2-quinolone, 7-amino-4,6-dimethyl-2-quinolone, 6-amino-7-chloro-4-methyl-2-quinolone, 7-amino-4-methyl-6-methoxy-2-quinolone, 5-aminobenzoxazolone, 6-amino-benzoxazolone, 6-amino-5-methyl-benzoxazolone, 6-amino-5-chloro-benzoxazolone, 6-amino-3-phenmorpholone, 7-amino-6-chloro-3-phenmorpholone, 7-amino-6-methyl-3-phenmorpholone, 7-amino-6-methoxy-3-phenmorpholone, 6-amino-4-methyl-3-phenmorpholone, 7-amino-4-methyl-3-phenmorpholone, 7-amino-4,6-dimethyl-3-phenmorpholone, 6-amino-4-quinazolinone and 5-aminophthalimide, and Y 1 is --H, OCH 3 , --OC 2 H 5 or --NHCOCH 3 , with the proviso that X 3 must not be H, if X is --O-- or --NH--.
Claim 2
Dependent Claim
363 words
A compound of the formulae I or II ##STR32## in which A is a radical of the formulae III, IV or V ##STR33## R 1 and R 4 are --H or --Cl, R 2 and R 5 are --H, halogen, --NO 2 , --CN, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, --CF 3 or phenyloxy which is unsubstituted or substituted by one or two chlorine atoms, one or two methyl or methoxy groups, or by one or two chlorine atoms and one or two methyl or methoxy groups and R 3 is alkyl having at least 10 C atoms, X is a radical of the formulae --NH--, --O--, ##STR34## n is the number 1 or 2, Y is the radical of the formulae --COO--, --OOC--, --CONH-- or --NHCO-- or a radical of the formulae ##STR35## in which R 1 and R 2 are as defined above, D is a 5-benzimidazolonyl, 5- or 6-benzoxazolonyl, 6-(2,4-dihydroxy)-quinazolinyl, 6- or 7-(4-methyl)quinolone-2-yl, 6- or 7-phenmorpholone-3-yl or 6-quinazolone-4-yl radical, Z is --H, --Br, --OCH 3 , --CN or --NO 2 and X 1 , and X 2 , independently of one another, are --H, halogen, --CH 3 , --OCH 3 --OC 2 H 5 or --NO 2 and X 3 is --H, --NHCO--C 1 -C 4 -alkyl, benzoylamino or phenylcarboxamido which are each unsubstituted or substituted on the phenyl ring by one or two chlorine atoms, one or two methyl or methoxy groups, one or two chlorine atoms and one or two methyl or methoxy groups, or an --NHCO--C 1 -C 4 alkyl group, or X 2 and X 3 together with the carbon atom to which they are bound are an aromatic carboxylic 6-membered ring or an aromatic heterocyclic 5- or 6-membered ring selected from the group consisting of 5-amino-benzimidazolone, 7-chloro-5-amino-benzimidazolone, 7-bromo-5-amino-benzimidazolone, 6-chloro-5-amino-benzimidazolone, 6-bromo-5-amino-benzimidazolone, 6-methoxy-5-amino-benzimidazolone, 7-methoxy-5-amino-benzimidazolone, 6-ethoxy-5-amino-benzimidazolone, 7-chloro-4-methyl-5-amino-benzimidazolone, 6-methyl-5-amino-benzimidazolone, 4,7-dimethyl-5-amino-benzimidazolone, 4-methyl-6-chloro-5-amino-benzimidazolone, 5-amino-1-methyl-benzimidazolone, 6-amino-2,4-dihydroxyquinazoline, 6-amino-1,4-dihydroxyquinazoline, 6-amino-4-methyl-2-quinolone, 7-amino-4-methyl-2-quinolone, 7-amino-4,6-dimethyl-2-quinolone, 6-amino-7-chloro-4-methyl-2-quinolone, 7-amino-4-methyl-6-methoxy-2-quinolone, 5-aminobenzoxazolone, 6-amino-benzoxazolone, 6-amino-5-methyl-benzoxazolone, 6-amino-5-chloro-benzoxazolone, 6-amino-3-phenmorpholone, 7-amino-6-chloro-3-phenmorpholone, 7-amino-6-methyl-3-phenmorpholone, 7-amino-6-methoxy-3-phenmorpholone, 6-amino-4-methyl-3-phenmorpholone, 7-amino-4-methyl-3-phenmorpholone, 7-amino-4,6-dimethyl-3-phenmorpholone, 6-amino-4-quinazolinone and 5-aminophthalimide, and Y 1 is --H, OCH 3 , --OC 2 H 5 or --NHCOCH 3 , with the proviso that X 3 must not be H, if X is --O-- or --NH--.
Claim 3
Dependent Claim
29 words
A compound according to claim 1, in which X is --O-- or --NH--, Y is a radical of the formula --COO-- or --CONH-- and n is the number 1.
Claim 4
Dependent Claim
27 words
A compound according to claim 1, in which R 3 is C 12 -C 35 alkyl, Y is --COO-- or --CONH-- and n is the number 1.
Claim 5
Dependent Claim
183 words
A compound according to claim 1, which has the formulae VI or VII ##STR36## in which X is --O-- or --NH--, R 1 is --H or --Cl, and R 2 is --Cl, --OCH 3 , --CH 3 , --OC 2 H 5 or --OC 6 H 5 , A is a radical of the formula III according to claim 12 in which Z is --H, X 1 and X 2 , independently of one another, are --H, --Cl, --CH 3 or --OCH 3 , and X 3 is --H, --NHCOCH 3 , benzoylamino or phenylcarboxamido which are each unsubstituted or substituted by one or two chlorine atoms, one or two methyl or methoxy groups, one or two chlorine atoms and one or two methyl or methoxy groups or by --NHCOCH 3 , or X 2 and X 3 together with the carbon atom to which they are bound form a ring of the formulae ##STR37## and R 3 is C 12 -C 18 alkyl, with the proviso that X 3 in formula VI must not be --H, if X is --O-- or --NH--.
Claim 6
Dependent Claim
41 words
A compound according to claim 4, in which R 1 is --H, R 2 is --Cl, --CH 3 or --OCH 3 , and the group --COXR 3 in formula VII is in the para-position relative to the group R 2 .
Claim 7
Dependent Claim
33 words
A compound according to claim 4, which has the formula VIII ##STR38## in which X is --O-- or --NH--, R 2 is --CH 3 and R 3 is C 12 -C 18 alkyl.
Claim 8
Dependent Claim
132 words
A compound according to claim 1, which has the formula IX or X ##STR39## in which X is --O--, or --NH--, R 1 is --H or --Cl, R 2 is --Cl, --CH 3 or --OCH 3 and R 3 is C 12 -C 18 alkyl, X 1 and X 2 , independently of one another, are --H, --Cl, --CH 3 or --OCH 3 , and X 3 is --H, --NHCOCH 3 , benzoylamino which is unsubstituted or substituted by one or two chlorine atoms, one or two methyl or methoxy groups, one or two chlorine atoms and one or two methyl or methoxy groups or by --NHCOCH 3 , or X 2 and X 3 together with the carbon atom to which they are bound form a ring of the formula ##STR40##
Claim 9
Dependent Claim
115 words
A compound of the formulae XI ##STR41## in which n is the number 1 or 2, R 1 is --H or --Cl, R 2 is --H, halogen, --NO 2 , --CN, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, --CF 3 or phenyloxy which is unsubstituted or substituted by one or two chlorine atoms, one or two methyl or methoxy groups, or one or two chlorine atoms and one or two methyl or methoxy groups, R 3 is alkyl having at least 10 C atoms, Z is --H, --Br, --OCH 3 , --CN or NO 2 , T is --OH or halogen and X is a radical of the formulae --NH--, --O--, ##STR42##
Claim 10
Dependent Claim
115 words
A compound of the formulae XI ##STR41## in which n is the number 1 or 2, R 1 is --H or --Cl, R 2 is --H, halogen, --NO 2 , --CN, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, --CF 3 or phenyloxy which is unsubstituted or substituted by one or two chlorine atoms, one or two methyl or methoxy groups, or one or two chlorine atoms and one or two methyl or methoxy groups, R 3 is alkyl having at least 10 C atoms, Z is --H, --Br, --OCH 3 , --CN or NO 2 , T is --OH or halogen and X is a radical of the formulae --NH--, --O--, ##STR42##
Claim 11
Dependent Claim
12 words
A compound according to claim 8, which has the formula XIII ##STR43##
Claim 12
Dependent Claim
45 words
A compound of the formula XIII according to claim 9, in which R 1 is --H, R 2 is --Cl, --CH 3 or --OCH 3 , R 3 is C 12 -C 18 alkyl, X is --O-- or --NH-- and T is --OH or --Cl.