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Controlled release compositions and their preparation

Assignee: Strong Cobb Arner Inc
•
Filing: 1961-04-28
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Granted: 1963-08-20
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Expires: 1981-04-28
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Abstract

No abstract record available.

Inventors

  • 👤 William E Gaunt
  • 👤 Robert P Tansey

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-10-24 22:30
CPC Classifications
A; A61; A61K; A61K9/00; A61K9/14; A61K9/16; A61K9/1605; A61K9/1629; A61K9/1652; A61K9/1617

Claims Analysis

Total Claims: 2
Claim 1
Independent Claim 116 words
A PROCESS FOR PREPARING A CONTROLLED RELEASE COMPOSITION WHICH REGULATES THE RATE OF RELEASE OF A THERAPEUTIC AGENT INTO ALIMENTARY FLUIDS VARYING IN PH FROM THE ACIDITY OF GASTRIC JUICE TO THE ALKALINITY OF INTESTINAL FLUIDS WHICH COMPRISES COMBINING A SOLUTION OF AN ACID-RESISTANT ALKALISUSCEPTIBLE MATERIAL IN A NON-POLAR/POLAR SOLVENT MIXTURE CONTAINING AT LEAST ABOUT 50% NON-POLAR SOLVENT WITH A SEPARATE SOLUTION OF AN ALKALI-RESISTANT ACID-SUCEPTIBLE MATERIAL IN THE SAME SOLVENT MIXTURE, INCORPORATING A THERAPEUTIC AGENT INTO ONE OF SAID SOLUTIONS PRIOR TO COMBINING THE SOLUTIONS, REMOVING SOLVENT FROM TE GEL STRUCTURE WHICH FORMS AND BREAKING THE DRIED GEL INTO PARTICLES, WHEREBY EACH GEL PARTICLE HAS THE THERAPEUTIC AGENT SUBSTANTIALLY UNIFORMLY DISPERSED THERETHROUGH IN DISCRETE FORM.
Claim 2
Dependent Claim 116 words
A PROCESS FOR PREPARING A CONTROLLED RELEASE COMPOSITION WHICH REGULATES THE RATE OF RELEASE OF A THERAPEUTIC AGENT INTO ALIMENTARY FLUIDS VARYING IN PH FROM THE ACIDITY OF GASTRIC JUICE TO THE ALKALINITY OF INTESTINAL FLUIDS WHICH COMPRISES COMBINING A SOLUTION OF AN ACID-RESISTANT ALKALISUSCEPTIBLE MATERIAL IN A NON-POLAR/POLAR SOLVENT MIXTURE CONTAINING AT LEAST ABOUT 50% NON-POLAR SOLVENT WITH A SEPARATE SOLUTION OF AN ALKALI-RESISTANT ACID-SUCEPTIBLE MATERIAL IN THE SAME SOLVENT MIXTURE, INCORPORATING A THERAPEUTIC AGENT INTO ONE OF SAID SOLUTIONS PRIOR TO COMBINING THE SOLUTIONS, REMOVING SOLVENT FROM TE GEL STRUCTURE WHICH FORMS AND BREAKING THE DRIED GEL INTO PARTICLES, WHEREBY EACH GEL PARTICLE HAS THE THERAPEUTIC AGENT SUBSTANTIALLY UNIFORMLY DISPERSED THERETHROUGH IN DISCRETE FORM.

References Cited (Backward Citations)

US2805977A Cited
US2928769A Cited
US2987445A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1966-08-19 1967-02-18 1967-08-20 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1970-08-19 1971-02-18 1971-08-20 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1974-08-19 1975-02-18 1975-08-20 $7700.00 Window Closed / Lapsed

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