US4057629A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Tyrosine derivatives and process for preparing the same
Assignee: Daiichi Pharmaceutical Co Ltd
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Filing: 1976-12-20
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Granted: 1977-11-08
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Expires: 1996-12-20
Abstract
Abstract Compounds having the formula: ##STR1## wherein R 1 is phenyl or cycloalkyl and the phenyl may have at least one substituent selected from the group consisting of lower alkyl, lower alkoxy, amino and nitro; R 2 is hydrogen or lower alkyl; A is --CH 2 O-- or --CH 2 CH(O-lower alkyl)-; n is zero (0) or one (1); when R 1 together with (A) n is unsubstituted phenyl, R 2 is lower alkyl; and R 3 is hydrogen or lower alkoxy, have anti-ulcerousaction.
Inventors
- 👤 Tosaku Miki
- 👤 Yasuhiro Hosokawa
- 👤 Tamotsu Miwa
- 👤 Hiroshi Fujita
- 👤 Masahide Asano
- 👤 Shunzo Aibara
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-10-30 11:32
CPC Classifications
C; C07; C07K; C07K5/00; C07K5/04; C07K5/06; C07K5/06191; C07K5/08; C07K5/0827; C07K5/10; C07K5/1027
Claims Analysis
Total Claims: 5
Claim 1
Independent Claim
19 words
The compound having the formula: ##STR18## wherein R 3 is hydrogen or a lower alkoxy, or a salt thereof.
Claim 2
Dependent Claim
19 words
The compound having the formula: ##STR18## wherein R 3 is hydrogen or a lower alkoxy, or a salt thereof.
Claim 3
Dependent Claim
9 words
The compound of claim 1 which is N-(4-methoxybenzoyl) phenylalanyltyrosine.
Claim 4
Dependent Claim
8 words
The compound of claim 1 which is N-benzoylphenylalanyltyrosine.
Claim 5
Dependent Claim
23 words
The method of treating ulcers in humans which comprises administering a compound of claim 1 in an amount effective for treating said ulcers.
References Cited (Backward Citations)
GB1201121A
Cited
US3778427A
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1980-11-07 | 1981-05-09 | 1981-11-08 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1984-11-07 | 1985-05-09 | 1985-11-08 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1988-11-07 | 1989-05-09 | 1989-11-08 | $7700.00 | Window Closed / Lapsed |